SCHEMBL28061207

SCHEMBL28061207

CC(C)[Si](C(C)C)(C(C)C)n1ccc2cncnc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK2 Q9HBH9 8/20 0.40
MKNK1 Q9BUB5 2/20 0.34
IRAK4 Q9NWZ3 5/20 0.33
EGFR P00533 4/20 0.32
PIK3CD O00329 4/20 0.32
PIK3CA P42336 4/20 0.32
PIK3CB P42338 4/20 0.32
MTOR P42345 4/20 0.32
PIK3CG P48736 4/20 0.32
ABL1 P00519 3/20 0.32
HCK P08631 3/20 0.32
SRC P12931 3/20 0.32
KDR P35968 3/20 0.32
EPHB4 P54760 3/20 0.32
PRKDC P78527 3/20 0.32
CYP1A2 P05177 2/20 0.31
CYP3A4 P08684 2/20 0.31
TSHR P16473 2/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6364432 0.75 MKNK2 (0.42) MKNK2MKNK1IRAK4EGFRPIK3CD
SCHEMBL417021 0.75 CCR1 (0.40) CYP1A2
SCHEMBL1883096 0.74 PARP1 (0.44) CYP2C19
SCHEMBL4478005 0.73 IRAK4 (0.34) IRAK4
SCHEMBL855838 0.73 HPGD (0.36) IRAK4TSHRALDH1A1
SCHEMBL5615371 0.73
SCHEMBL256370 0.72 MKNK2 (0.45) MKNK2MKNK1EGFRPIK3CBCYP1A2
SCHEMBL30694603 0.72 MKNK2 (0.45) MKNK2MKNK1EGFRPIK3CBCYP1A2
SCHEMBL18926936 0.71 MKNK2 (0.39) MKNK2MKNK1IRAK4
SCHEMBL29533363 0.71 HTR2C (0.35) EGFRABL1HCKSRCCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103732597-B Tricyclic heterocyclic compounds and JAK inhibitors 日产化学工业株式会社 2016-08-17 CN disclosed