SCHEMBL28061209

SCHEMBL28061209

O=c1cc[nH]c2c1cnc1[nH]cnc12

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR8 P51685 1/20 0.46
KMT2A Q03164 1/20 0.44
CHEK1 O14757 1/20 0.37
ADORA2A P29274 2/20 0.37
ADORA1 P30542 1/20 0.37
PARP1 P09874 5/20 0.36
IGF1R P08069 2/20 0.36
PIM1 P11309 2/20 0.36
CLK2 P49760 2/20 0.36
GSK3A P49840 2/20 0.36
GSK3B P49841 2/20 0.36
DYRK1A Q13627 2/20 0.36
CLK4 Q9HAZ1 2/20 0.36
AURKA O14965 1/20 0.36
DAPK3 O43293 1/20 0.36
JAK2 O60674 1/20 0.36
PRKD3 O94806 1/20 0.36
MAP4K4 O95819 1/20 0.36
PAK4 O96013 1/20 0.36
ABL1 P00519 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14697441 0.79 CCR8 (0.52) CCR8KMT2AADORA2AADORA1DYRK1A
SCHEMBL17353634 0.66 PRKCI (0.42) CHEK1DYRK1AJAK2JAK3AXL
SCHEMBL12540118 0.65 ABL1 (0.48) CCR8KMT2AADORA2AADORA1ABL1
SCHEMBL30774416 0.65 CCR8 (1.00) CCR8KMT2AADORA2AADORA1PARP1
SCHEMBL22643575 0.65 CCR8 (0.43) CCR8KMT2AADORA2AADORA1BTK
SCHEMBL19318056 0.65 CCR8 (1.00) CCR8KMT2AADORA2AADORA1PARP1
SCHEMBL2211844 0.64 CCR8 (0.42) CCR8KMT2AADORA2AADORA1SMN1; SMN2
SCHEMBL20887679 0.63 CCR8 (0.50) CCR8KMT2AADORA2AADORA1PARP1
SCHEMBL19012489 0.63 CCR8 (0.50) CCR8KMT2AADORA2AADORA1PARP1
SCHEMBL31300928 0.62 TET2 (0.55) CCR8KMT2AADORA2AADORA1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103732597-B Tricyclic heterocyclic compounds and JAK inhibitors 日产化学工业株式会社 2016-08-17 CN disclosed