SCHEMBL28066688

SCHEMBL28066688

CCCCCc1cccnc1C(=O)OCC

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.53
TDP2 O95551 2/20 0.43
CYP4F2 P78329 1/20 0.43
CYP4A11 Q02928 1/20 0.43
PDE4A P27815 1/20 0.42
PPARA Q07869 3/20 0.41
LMNA P02545 1/20 0.41
KDM4E B2RXH2 1/20 0.41
KDM4A O75164 1/20 0.41
KDM4C Q9H3R0 1/20 0.41
CYP1A2 P05177 1/20 0.41
BID P55957 3/20 0.40
MCL1 Q07820 3/20 0.40
BCL2L1 Q07817 2/20 0.40
BAK1 Q16611 2/20 0.40
KAT8 Q9H7Z6 2/20 0.40
PPARG P37231 2/20 0.40
EP300 Q09472 1/20 0.40
KAT2A Q92830 1/20 0.40
KAT2B Q92831 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28472394 0.85 BRD4 (0.61) BRD4TDP2PDE4ALMNAKDM4E
SCHEMBL14895437 0.84 BRD4 (0.58) BRD4TDP2PDE4ALMNAKDM4E
SCHEMBL5498415 0.82 KDM4E (0.58) PPARAKDM4ECYP1A2BIDMCL1
SCHEMBL18598998 0.82 BID (0.44) PPARAKDM4ECYP1A2BIDMCL1
SCHEMBL10932980 0.82 BID (0.44) PPARAKDM4ECYP1A2BIDMCL1
SCHEMBL18132204 0.82 BRD4 (0.58) BRD4TDP2CYP4F2CYP4A11PDE4A
SCHEMBL24908480 0.81 KDM4E (0.57) PPARAKDM4ECYP1A2BIDMCL1
SCHEMBL3369457 0.81 BRD4 (0.57) BRD4TDP2PDE4AKDM4ECYP1A2
SCHEMBL9094733 0.81 KDM4E (0.57) PPARAKDM4ECYP1A2BIDMCL1
SCHEMBL7908951 0.81 BRD4 (0.57) BRD4TDP2PDE4AKDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109053742-A New tricyclic compound ABBVIE 公司 2018-12-21 CN disclosed
CN-106046106-A C-3 cycloalkenyl triterpenoids with HIV maturation inhibitory activity 百时美施贵宝公司 2016-10-26 CN disclosed
CN-104220451-B C-3 cycloalkene triterpenoids with HIV maturation inhibitory activity 百时美施贵宝公司 2016-06-29 CN disclosed