SCHEMBL28069573

SCHEMBL28069573

Cn1c(=O)cc(N2CCC[C@@H](NC(=O)OC(C)(C)C)C2)n(Cc2cc(F)ccc2C#N)c1=O

nearest known ligand 0.68

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 19/20 0.68
OPRM1 P35372 1/20 0.53
OPRK1 P41145 1/20 0.53
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
RET P07949 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28507242 1.00 DPP4 (0.68) DPP4OPRM1OPRK1CYP1A2CYP3A4
SCHEMBL13185937 0.90 DPP4 (0.66) DPP4OPRM1OPRK1
SCHEMBL17781891 0.90 DPP4 (0.66) DPP4OPRM1OPRK1
SCHEMBL16280698 0.85 DPP4 (0.72) DPP4CYP1A2CYP3A4CYP2D6RET
SCHEMBL28324302 0.83 DPP4 (0.69) DPP4RET
SCHEMBL2022448 0.82 DPP4 (0.69) DPP4RET
SCHEMBL2022446 0.82 DPP4 (0.69) DPP4RET
SCHEMBL10331078 0.82 DPP4 (0.84) DPP4OPRM1OPRK1CYP1A2CYP3A4
SCHEMBL13141899 0.82 DPP4 (0.84) DPP4OPRM1OPRK1CYP1A2CYP3A4
SCHEMBL18851350 0.81 DPP4 (0.67) DPP4RET

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646447-A Synthesis method of dipeptidyl peptidase inhibitor 北京康立生医药技术开发有限公司 2016-06-08 CN disclosed