SCHEMBL28072254

SCHEMBL28072254

BrN1CCC(c2cnccn2)C1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 1/20 0.42
EPHX2 P34913 1/20 0.42
MAP4K4 O95819 1/20 0.41
PDCD1LG2 Q9BQ51 1/20 0.40
CD274 Q9NZQ7 1/20 0.40
NAMPT P43490 1/20 0.40
CHRM2 P08172 3/20 0.36
CHRM1 P11229 3/20 0.36
HRH3 Q9Y5N1 1/20 0.36
PRMT5 O14744 1/20 0.34
WDR77 Q9BQA1 1/20 0.34
CHRM4 P08173 2/20 0.33
CHRM5 P08912 2/20 0.33
CHRM3 P20309 2/20 0.33
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13123169 0.82 CYP2C9 (0.40) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL19087064 0.82 PDCD1LG2 (0.41) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL7920351 0.82 PDCD1LG2 (0.41) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL19116698 0.80 CD274 (0.47) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL19077886 0.78 CYP2C9 (0.41) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL6232040 0.78 KDM4E (0.38) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL28262276 0.78 MAP4K4 (0.39) CYP2C9EPHX2MAP4K4PDCD1LG2CD274
SCHEMBL14250161 0.78
SCHEMBL30339210 0.78
SCHEMBL12090384 0.76 MAP4K4 (0.46) CYP2C9EPHX2MAP4K4CHRM2CHRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105622526-A Preparation method of 2-aminopyrazine derivatives UNIV HUBEI TECHNOLOGY 2016-06-01 CN claimed
CN-105622526-A Preparation method of 2-aminopyrazine derivatives UNIV HUBEI TECHNOLOGY 2016-06-01 CN disclosed