SCHEMBL28075797

SCHEMBL28075797

O=C(Nc1cnccc1-c1ccc(F)cc1)c1cnccn1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3A P49840 10/20 0.66
GSK3B P49841 9/20 0.66
JAK2 O60674 2/20 0.66
PIM1 P11309 2/20 0.66
CDK2 P24941 2/20 0.66
CDK5 Q00535 2/20 0.66
PRKCQ Q04759 2/20 0.66
AURKB Q96GD4 2/20 0.66
TYK2 P29597 1/20 0.66
SYK P43405 1/20 0.66
TSHR P16473 2/20 0.62
ALDH1A1 P00352 1/20 0.62
ALOX15 P16050 1/20 0.62
MEN1 O00255 1/20 0.58
CDC25A P30304 1/20 0.58
CDC25B P30305 1/20 0.58
CDC25C P30307 1/20 0.58
HTT P42858 1/20 0.58
KMT2A Q03164 1/20 0.58
IGF1R P08069 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28125970 0.84 TSHR (0.56) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL29939262 0.83 GSK3A (0.74) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL20204912 0.83 GSK3A (0.74) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL20205153 0.80 GSK3A (1.00) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL29939440 0.80 GSK3A (1.00) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL28075793 0.80 GSK3A (0.61) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL16703316 0.79 GSK3B (0.67) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL20204929 0.77 GSK3A (0.76) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL29939337 0.77 GSK3A (0.76) GSK3AGSK3BJAK2PIM1CDK2
SCHEMBL29939261 0.77 GSK3A (1.00) GSK3AGSK3BJAK2PIM1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849098-A Gsk-3 inhibitors 百时美施贵宝公司 2016-08-10 CN disclosed