SCHEMBL28076877

SCHEMBL28076877

CC1(C)Cc2ccc(-c3ccc(CN)cc3)cc2O1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 1/20 0.42
TAAR1 Q96RJ0 4/20 0.39
CD274 Q9NZQ7 1/20 0.39
PIM1 P11309 1/20 0.38
PIM3 Q86V86 1/20 0.38
PIM2 Q9P1W9 1/20 0.38
KIT P10721 1/20 0.37
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
HIF1A Q16665 4/20 0.34
EPAS1 Q99814 4/20 0.34
MET P08581 1/20 0.33
MAOB P27338 1/20 0.32
HTR2A P28223 1/20 0.32
CYP2A6 P11509 1/20 0.32
CTSD P07339 1/20 0.32
BACE1 P56817 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL660552 0.81 KIT (0.41) PIM1PIM3PIM2KITMET
SCHEMBL13156334 0.78 HIF1A (0.44) HIF1AEPAS1MAOBHTR2A
SCHEMBL15599255 0.76 PARP1 (0.37) PIM1PIM3PIM2HIF1AEPAS1
SCHEMBL11358788 0.74 CNR2 (0.38) HIF1AEPAS1MAOB
SCHEMBL18053881 0.72 MAPT (0.41) PIM1PIM3PIM2
SCHEMBL30781068 0.72 MAPT (0.41) PIM1PIM3PIM2
SCHEMBL30523622 0.71 MAOB (0.35) PIM1PIM3PIM2HIF1AEPAS1
SCHEMBL660359 0.71 CYP11B1 (0.52) CYP2A6CTSDBACE1
SCHEMBL8959298 0.70 AKR1B1 (0.43) HIF1A
SCHEMBL12180466 0.70 KDM4E (0.38) PIM1PIM3PIM2KITMAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103965147-B Benzofuran derivatives 武田药品工业株式会社 2016-08-24 CN disclosed