SCHEMBL28077563

SCHEMBL28077563

O=CC1(COCc2ccccc2)CCN(C(=O)O)CC1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 4/20 0.42
MEN1 O00255 2/20 0.41
KMT2A Q03164 2/20 0.41
NPSR1 Q6W5P4 1/20 0.41
TEAD3 Q99594 1/20 0.41
TACR1 P25103 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
CYP2D6 P10635 2/20 0.40
USP2 O75604 1/20 0.40
ALDH1A1 P00352 1/20 0.40
CYP3A4 P08684 1/20 0.40
MAPK1 P28482 1/20 0.40
CYP2C19 P33261 2/20 0.39
SLC1A3 P43003 2/20 0.38
SLC1A2 P43004 2/20 0.38
SLC1A1 P43005 2/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16554179 0.85 TACR1 (0.55) MEN1KMT2ATACR1
SCHEMBL6170590 0.84 TSHR (0.48) MEN1KMT2ATACR1CYP2D6ALDH1A1
SCHEMBL100117 0.81 TACR1 (0.45) MEN1KMT2ATACR1CYP2D6ALDH1A1
SCHEMBL28654159 0.81 TACR1 (0.45) MEN1KMT2ATACR1CYP2D6ALDH1A1
SCHEMBL30195760 0.81 TACR1 (0.51) TACR1HDAC1HDAC6
SCHEMBL16554180 0.79 GRM5 (0.35) GRM5TACR1SMN1; SMN2NPC1RAB9A
SCHEMBL7713336 0.78 TACR1 (0.42) GRM5MEN1KMT2ANPSR1TACR1
SCHEMBL28831286 0.78 GRM5 (0.42) GRM5MEN1KMT2ANPSR1TEAD3
SCHEMBL26704597 0.78 TACR1 (0.40) MEN1KMT2ATEAD3TACR1SMN1; SMN2
SCHEMBL26704618 0.78 TACR1 (0.40) MEN1KMT2ATEAD3TACR1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105745209-A Triazolopyridine compounds, compositions, and methods of use thereof 豪夫迈·罗氏有限公司 2016-07-06 CN disclosed