SCHEMBL28079390

SCHEMBL28079390

Cc1cccc2nc(-c3ccccc3)c(-c3ccc4ccccc4c3)nc12

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.51
TDP1 Q9NUW8 2/20 0.50
ADORA2A P29274 3/20 0.49
ADORA1 P30542 3/20 0.49
MAPT P10636 1/20 0.48
MAPK1 P28482 1/20 0.48
RAB9A P51151 1/20 0.48
L3MBTL1 Q9Y468 4/20 0.46
KDM4E B2RXH2 4/20 0.46
LMNA P02545 4/20 0.46
ALDH1A1 P00352 3/20 0.46
NPSR1 Q6W5P4 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
GAA P10253 1/20 0.42
THRB P10828 1/20 0.42
DHODH Q02127 1/20 0.41
AKT1 P31749 1/20 0.41
AKT2 P31751 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12578244 0.87 MAPT (0.58) PDE10ATDP1MAPTMAPK1RAB9A
SCHEMBL11947016 0.84 PDE10A (0.44) PDE10ATDP1ADORA2AADORA1MAPT
SCHEMBL28079530 0.82 ADORA2A (0.62) PDE10ATDP1ADORA2AADORA1L3MBTL1
SCHEMBL12207312 0.79 TDP1 (0.50) PDE10ATDP1MAPTMAPK1RAB9A
SCHEMBL21667459 0.79 ADORA2A (0.46) PDE10ATDP1ADORA2AADORA1L3MBTL1
SCHEMBL12207290 0.79 TDP1 (0.50) PDE10ATDP1MAPTMAPK1RAB9A
SCHEMBL4750618 0.78 TDP1 (0.49) PDE10ATDP1MAPTMAPK1RAB9A
SCHEMBL22186546 0.78 ADORA2A (0.44) PDE10ATDP1ADORA2AADORA1MAPK1
SCHEMBL13614825 0.78 MAPT (0.47) PDE10ATDP1MAPTMAPK1RAB9A
SCHEMBL8802391 0.78 MAPT (0.51) PDE10ATDP1ADORA2AMAPTMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105693632-B A kind of preparation method of polysubstituted quinoxaline derivant 华侨大学 2018-04-17 CN disclosed
CN-105693632-A Preparation method of polysubstitution quinoxalin derivatives 华侨大学 2016-06-22 CN disclosed