SCHEMBL28079746

SCHEMBL28079746

NCC1(COCc2ccccc2)CCCN(C=O)C1

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 3/20 0.37
CYP2D6 P10635 5/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 4/20 0.35
CYP3A4 P08684 4/20 0.35
CXCR3 P49682 1/20 0.35
LTA4H P09960 1/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
USP2 O75604 1/20 0.34
GAA P10253 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SLC6A4 P31645 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5722244 0.80 TSHR (0.47) TACR1ALDH1A1TSHRCYP1A2USP2
SCHEMBL17100019 0.72 TSHR (0.52) TACR1TSHRLTA4H
SCHEMBL6127863 0.69 NPC1 (0.51) CYP2D6CYP3A4CYP1A2CYP2C9CYP2C19
SCHEMBL1981994 0.69 TACR1 (0.56) TACR1TSHR
SCHEMBL31721404 0.69 TACR1 (0.41) TACR1TSHRCYP2C9CYP2C19GAA
SCHEMBL19074506 0.68 TSHR (0.47) TACR1TSHRLTA4HSLC6A4
SCHEMBL3490325 0.68 TSHR (0.47) TACR1ALDH1A1TSHRGAANPC1
SCHEMBL6124701 0.68 SMN1; SMN2 (0.47) CYP2C19NPC1RAB9ASMN1; SMN2
SCHEMBL15043681 0.67 TACR1 (0.45) TACR1TSHRLTA4HSLC6A4
SCHEMBL28654159 0.67 TACR1 (0.45) TACR1CYP2D6ALDH1A1TSHRLTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105646532-A Synthesis method of 2-tertbutyloxycarbonyl-10-carbonyl-8-oxo-2,11-diazaspiro[5.6]dodecane 上海药明康德新药开发有限公司 2016-06-08 CN claimed
CN-105646532-A Synthesis method of 2-tertbutyloxycarbonyl-10-carbonyl-8-oxo-2,11-diazaspiro[5.6]dodecane 上海药明康德新药开发有限公司 2016-06-08 CN disclosed