SCHEMBL28080574

SCHEMBL28080574

CCCCCCC(Cc1ccccn1)C(N)=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.46
FDPS P14324 1/20 0.42
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
HPGD P15428 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HDAC6 Q9UBN7 5/20 0.40
HDAC1 Q13547 2/20 0.40
ALOX12 P18054 1/20 0.40
CTSK P43235 1/20 0.40
LPAR3 Q9UBY5 1/20 0.40
CYP1A2 P05177 2/20 0.40
GRIN2D O15399 1/20 0.40
GRIN3B O60391 1/20 0.40
GRIN1 Q05586 1/20 0.40
GRIN2A Q12879 1/20 0.40
GRIN2B Q13224 1/20 0.40
GRIN2C Q14957 1/20 0.40
GRIN3A Q8TCU5 1/20 0.40
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2134795 0.88 PTPRA (0.47) PTPRAFDPSHPGDHSD17B10HDAC6
SCHEMBL2187235 0.82 PTPRA (0.59) PTPRAFDPSCYP1A2GRIN2DGRIN3B
SCHEMBL7789683 0.79 CSNK1E (0.57) CSNK1E
SCHEMBL22558568 0.79 CSNK1E (0.57) CSNK1E
SCHEMBL28058533 0.79 CSNK1E (0.57) CSNK1E
SCHEMBL28081007 0.79 CSNK1E (0.57) CSNK1E
SCHEMBL22118359 0.79 GRIN2D (0.49) PTPRAFDPSALOX12GRIN2DGRIN3B
SCHEMBL1532579 0.79 PTPRA (0.47) PTPRAFDPSHPGDHSD17B10ALOX12
SCHEMBL21770640 0.78 GRIN2D (0.44) PTPRAFDPSALOX12GRIN2DGRIN3B
SCHEMBL29058174 0.78 GRIN2D (0.44) PTPRAFDPSALOX12GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106967066-B Novel ss-lactam enzyme inhibitor and preparation method thereof 明治制果药业株式会社 2019-07-30 CN disclosed
CN-105859609-B Beta-lactamase inhibitor and preparation method thereof 明治制果药业株式会社 2019-04-09 CN disclosed
CN-106967066-A New beta lactamase restrainer and preparation method thereof 明治制果药业株式会社 2017-07-21 CN disclosed
CN-104334559-B Beta-lactamase inhibitor and preparation method thereof 明治制果药业株式会社 2017-03-22 CN disclosed
CN-105859609-A Beta-lactamase inhibitor and process for preparing the same 明治制果药业株式会社 2016-08-17 CN disclosed