SCHEMBL28080965

SCHEMBL28080965

CC(N)c1cnc(OCC(F)(F)C(F)F)c(Cl)c1

nearest known ligand 0.42

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 10/20 0.42
MAPK1 P28482 1/20 0.39
AAK1 Q2M2I8 5/20 0.37
IDH1 O75874 4/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL15350461 0.99 SCN9A (0.42) SCN9AMAPK1AAK1IDH1
SCHEMBL17244897 0.89 SCN9A (0.42) SCN9AMAPK1AAK1IDH1
SCHEMBL16045149 0.87 IDH1 (0.43) SCN9AAAK1IDH1
SCHEMBL4550317 0.87 IDH1 (0.43) SCN9AAAK1IDH1
Hydrochloric Acid SCHEMBL2714340 0.86 IDH1 (0.43) SCN9AAAK1IDH1
SCHEMBL10291359 0.85 MAPK1 (0.42) SCN9AMAPK1AAK1
Hydrochloric Acid SCHEMBL15350476 0.85 AAK1 (0.40) AAK1IDH1
Hydrochloric Acid SCHEMBL2717390 0.84 MAPK1 (0.41) SCN9AMAPK1AAK1
SCHEMBL18266454 0.80 SCN9A (0.34) SCN9AAAK1
SCHEMBL4550399 0.80 SCN9A (0.39) SCN9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104520296-B Pyrrolopyridinone derivatives as TTX-S blocker 拉夸里亚创药株式会社 2016-11-16 CN disclosed