SCHEMBL28080986

SCHEMBL28080986

CC(F)(F)COc1ncccc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SSTR4 P31391 4/20 0.46
NFE2L2 Q16236 2/20 0.38
HDAC1 Q13547 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
HDAC5 Q9UQL6 1/20 0.36
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
ATM Q13315 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
NUDT1 P36639 1/20 0.35
MKNK1 Q9BUB5 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
GAA P10253 1/20 0.35
SCN9A Q15858 1/20 0.34
SSTR1 P30872 1/20 0.34
RXRA P19793 1/20 0.34
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
TRPV4 Q9HBA0 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10324235 0.90 SSTR4 (0.46) SSTR4NFE2L2HDAC1HDAC6HDAC5
SCHEMBL16174985 0.86 SSTR4 (0.42) SSTR4HDAC1HDAC6HDAC5KMT2A
SCHEMBL16239660 0.83 SSTR4 (0.41) SSTR4NFE2L2HDAC1HDAC6HDAC5
SCHEMBL24599918 0.80 SSTR4 (0.39) SSTR4NFE2L2HDAC1HDAC6HDAC5
SCHEMBL364602 0.80 SSTR4 (0.39) SSTR4HDAC1HDAC6HDAC5KMT2A
SCHEMBL24599912 0.79 SSTR4 (0.39) SSTR4NFE2L2HDAC1HDAC6HDAC5
SCHEMBL24599915 0.78 SSTR4 (0.38) SSTR4HDAC1HDAC6HDAC5ALDH1A1
SCHEMBL24599913 0.78 SSTR4 (0.38) SSTR4HDAC1HDAC6HDAC5ALDH1A1
SCHEMBL24599855 0.78 SSTR4 (0.38) SSTR4HDAC1HDAC6HDAC5ALDH1A1
SCHEMBL16175292 0.76 EPHX2 (0.39) SSTR4HDAC1HDAC6HDAC5ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104520296-B Pyrrolopyridinone derivatives as TTX-S blocker 拉夸里亚创药株式会社 2016-11-16 CN disclosed