SCHEMBL28089341

SCHEMBL28089341

CC(C)c1cc(CCOC=O)n[nH]1

nearest known ligand 0.39

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 2/20 0.39
HCAR3 P49019 1/20 0.39
PRKAB2 O43741 5/20 0.34
PRKAG1 P54619 5/20 0.34
PRKAA2 P54646 5/20 0.34
PRKAA1 Q13131 5/20 0.34
PRKAG3 Q9UGI9 5/20 0.34
PRKAG2 Q9UGJ0 5/20 0.34
PRKAB1 Q9Y478 5/20 0.34
CCNA2 P20248 1/20 0.33
CDK2 P24941 1/20 0.33
CCNA1 P78396 1/20 0.33
KDM5A P29375 6/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
KDM5B Q9UGL1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28391037 0.88 KDM5A (0.31) HCAR2HCAR3KDM5A
SCHEMBL27934105 0.77 HCAR2 (0.32) HCAR2
SCHEMBL27627220 0.76 HCAR2 (0.31) HCAR2
SCHEMBL28035629 0.76
SCHEMBL28289418 0.75 STK25 (0.36) NPC1RAB9ASMN1; SMN2
SCHEMBL28327146 0.75
SCHEMBL28888382 0.74 MAPK1 (0.32) HCAR2HCAR3
SCHEMBL27413353 0.73 HCAR2 (0.41) HCAR2
SCHEMBL10401170 0.72
SCHEMBL27758189 0.72 HCAR2 (0.38) HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106255688-B Morpholine-pyridine derivate 豪夫迈·罗氏有限公司 2019-11-08 CN disclosed
CN-106255688-A Morpholine pyridine derivate 豪夫迈·罗氏有限公司 2016-12-21 CN disclosed
CN-104080787-B Pyrazolo pyrrolidine compound 诺华股份有限公司 2016-09-14 CN disclosed