SCHEMBL28095339

SCHEMBL28095339

CC(C)(C)OC(=O)Nc1ccc(CNC(F)(F)F)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 2/20 0.54
AURKA O14965 1/20 0.48
RPS6KB1 P23443 1/20 0.48
NAMPT P43490 2/20 0.48
DRD2 P14416 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
MAPK14 Q16539 1/20 0.46
HDAC1 Q13547 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
PPARG P37231 2/20 0.43
PSMB8 P28062 1/20 0.43
PPARA Q07869 1/20 0.43
MAPKAPK2 P49137 2/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
HDAC3 O15379 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17744946 0.88 CYP17A1 (0.57) CYP17A1AURKARPS6KB1NAMPTDRD2
SCHEMBL23336325 0.83 CYP17A1 (0.62) CYP17A1AURKARPS6KB1NAMPTDRD2
SCHEMBL31016329 0.82 CYP17A1 (0.57) CYP17A1AURKARPS6KB1NAMPTDRD2
SCHEMBL1853151 0.82 CYP17A1 (0.54) CYP17A1NAMPTHDAC1HDAC6PPARG
SCHEMBL132701 0.81 CYP17A1 (0.76) CYP17A1NAMPTDRD2PTGDR2MAPK14
SCHEMBL16523129 0.81 CYP17A1 (0.56) CYP17A1AURKARPS6KB1NAMPTDRD2
SCHEMBL13055402 0.80 CYP17A1 (0.59) CYP17A1NAMPTDRD2PTGDR2MAPK14
SCHEMBL15996891 0.80 SMN1; SMN2 (0.53) CYP17A1AURKARPS6KB1NAMPTDRD2
SCHEMBL6195004 0.80 CYP17A1 (0.61) CYP17A1AURKARPS6KB1NAMPTDRD2
SCHEMBL10361607 0.80 CYP17A1 (0.61) CYP17A1NAMPTDRD2PTGDR2MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105899496-A OXAZOLIDINONE DERIVATIVES AS PPAR LIGANDS 安达卢西亚健康服务部 2016-08-24 CN disclosed