SCHEMBL28098646

SCHEMBL28098646

COc1cc2c(N)ncnn2c1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
MAP4K4 O95819 3/20 0.43
KIT P10721 4/20 0.43
XDH P47989 1/20 0.36
PI4KA P42356 2/20 0.35
PI4K2B Q8TCG2 2/20 0.35
PI4K2A Q9BTU6 2/20 0.35
PI4KB Q9UBF8 2/20 0.35
NOS3 P29474 1/20 0.34
NOS1 P29475 1/20 0.34
NOS2 P35228 1/20 0.34
FGFR1 P11362 3/20 0.33
CLK1 P49759 1/20 0.33
ABL1 P00519 1/20 0.33
EGFR P00533 1/20 0.33
CDK1 P06493 1/20 0.33
SRC P12931 1/20 0.33
ABL2 P42684 1/20 0.33
RIPK2 O43353 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL275263 0.77 MAP4K4 (0.47) MAP4K4KITXDHPI4KAPI4K2B
SCHEMBL17074794 0.76 ACVR2A (0.37) MAP4K4XDHPI4KAPI4K2BPI4K2A
SCHEMBL15023106 0.76 KIT (0.43) MAP4K4KITFGFR1
SCHEMBL13075093 0.73 MAP4K4 (0.47) MAP4K4KIT
SCHEMBL19698007 0.73 MAP4K4 (0.47) MAP4K4KITPI4KAPI4K2BPI4K2A
SCHEMBL12173491 0.72 MAP4K4 (0.43) MAP4K4KITPI4KAPI4K2BPI4K2A
SCHEMBL23029838 0.70 ACVR2A (0.38) MAP4K4FGFR1CDK1
SCHEMBL12173489 0.70 KIT (0.44) MAP4K4KIT
SCHEMBL276566 0.70 KIT (0.44) MAP4K4KITFGFR1
SCHEMBL275845 0.69 MAP4K4 (0.52) MAP4K4KITPI4KBFGFR1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104245700-B Dibasic benzothienyl-pyrrolo-triazine and the purposes as FGFR inhibitors of kinases thereof 拜耳制药股份公司 2016-11-16 CN disclosed