SCHEMBL28100577

SCHEMBL28100577

COC(=O)c1nc2cccc(F)c2c(C(=O)OC)c1F

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TACR3 P29371 1/20 0.43
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
PARP1 P09874 1/20 0.39
ALDH1A1 P00352 4/20 0.39
KDM4E B2RXH2 3/20 0.39
FYN P06241 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HPGD P15428 2/20 0.38
ATM Q13315 1/20 0.38
MMP13 P45452 1/20 0.37
BDKRB1 P46663 1/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28100578 0.92 TACR3 (0.44) TACR3MEN1KMT2APARP1ALDH1A1
SCHEMBL1070351 0.72 CA12 (0.61) CA12CA1CA2CA7CA9
SCHEMBL9384941 0.71 MAPT (0.43) CA12CA1CA2CA7CA9
SCHEMBL8574143 0.71 CA12 (0.45) CA12CA1CA2CA7CA9
SCHEMBL16832920 0.71 NQO2 (0.54) KMT2APARP1KDM4EATMMMP13
SCHEMBL2862825 0.71 KDM4E (0.59) KDM4ESMN1; SMN2MAPT
SCHEMBL8573902 0.70 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL8569654 0.70 POLB (0.45) CA12CA1CA2CA7CA9
SCHEMBL8574343 0.70 CA12 (0.44) CA12CA1CA2CA7CA9
SCHEMBL10925688 0.70 SMN1; SMN2 (0.37) MEN1KMT2AALDH1A1KDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106029647-A Glucose transport inhibitors 拜耳制药股份公司 2016-10-12 CN disclosed