SCHEMBL28100731

SCHEMBL28100731

CC(C)(C)OC(=O)c1ccc(C[C@H](C(=O)O)c2ccc(Br)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
SLC7A5 Q01650 1/20 0.43
MME P08473 3/20 0.43
PTGS1 P23219 2/20 0.42
PTGS2 P35354 2/20 0.42
CYP2C9 P11712 2/20 0.40
CYP2C19 P33261 1/20 0.40
ESR1 P03372 3/20 0.39
ESR2 Q92731 2/20 0.39
KDM4E B2RXH2 2/20 0.39
MAPT P10636 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
PPARG P37231 3/20 0.38
EPHX2 P34913 1/20 0.38
PPARA Q07869 2/20 0.38
PPARD Q03181 1/20 0.38
CA12 O43570 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1921149 1.00 KMT2A (0.44) KMT2ACTSSCTSKSLC7A5MME
SCHEMBL1921150 1.00 KMT2A (0.44) KMT2ACTSSCTSKSLC7A5MME
SCHEMBL13494499 0.88 SLC7A5 (0.44) SLC7A5PTGS1PTGS2CYP2C9CYP2C19
SCHEMBL17338896 0.88 ESRRG (0.37) KMT2ACTSSCTSKSLC7A5MME
SCHEMBL17338899 0.88 ESRRG (0.37) KMT2ACTSSCTSKSLC7A5MME
SCHEMBL1919196 0.88 ESR1 (0.56) KMT2ACTSSCTSKSLC7A5MME
SCHEMBL23306974 0.85 ESR1 (0.44) KMT2ACTSSCTSKSLC7A5MME
SCHEMBL13494459 0.85 SLC7A5 (0.48) CTSSCTSKSLC7A5MMEALDH1A1
SCHEMBL1919093 0.85 SLC7A5 (0.48) CTSSCTSKSLC7A5MMEALDH1A1
SCHEMBL1918994 0.85 ESR1 (0.48) KMT2APTGS1PTGS2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107428682-B Amide derivatives, preparation method and medical application thereof 浙江海正药业股份有限公司 2021-02-02 CN disclosed
CN-107428682-A Amide derivatives, its preparation method and its purposes in medicine 浙江海正药业股份有限公司 2017-12-01 CN disclosed
CN-106336387-A Amides derivative, preparation method thereof and purpose of amides derivative on medicine 浙江海正药业股份有限公司 2017-01-18 CN disclosed