SCHEMBL28114095

SCHEMBL28114095

FC(F)n1ccc(-c2ccccc2)n1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.53
CYP19A1 P11511 1/20 0.37
RAB9A P51151 5/20 0.37
MEN1 O00255 2/20 0.37
KDM4E B2RXH2 5/20 0.36
HSD17B10 Q99714 4/20 0.36
NPC1 O15118 4/20 0.36
HPGD P15428 4/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
NTRK1 P04629 1/20 0.35
MAPT P10636 6/20 0.35
ALOX15 P16050 1/20 0.35
MAPK1 P28482 1/20 0.35
MCL1 Q07820 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2453561 0.83 KMT2A (0.57) KMT2ACYP19A1RAB9AMEN1KDM4E
SCHEMBL12777940 0.80 KMT2A (0.59) KMT2ACYP19A1RAB9AMEN1KDM4E
SCHEMBL2766811 0.77 KMT2A (0.50) KMT2ACYP19A1RAB9AMEN1KDM4E
SCHEMBL21323392 0.77 KMT2A (0.55) KMT2ACYP19A1RAB9AMEN1KDM4E
SCHEMBL18191174 0.77 KMT2A (0.50) KMT2ACYP19A1MEN1KDM4EHSD17B10
SCHEMBL20456867 0.77 DRD1 (0.41) KMT2AKDM4EHSD17B10ALDH1A1MAPK1
SCHEMBL23034625 0.74 KMT2A (0.52) KMT2ACYP19A1RAB9AMEN1KDM4E
Butadiene SCHEMBL2765437 0.74 KMT2A (0.47) KMT2ACYP19A1RAB9AMEN1KDM4E
SCHEMBL31457967 0.73 FYN (0.33) KMT2AMEN1LMNANTRK1MAPT
SCHEMBL17261541 0.73 KMT2A (0.50) KMT2ARAB9AKDM4ENPC1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104114555-B Pyrazolopyrimidine derivatives, process for their preparation and their therapeutic use 赛诺菲 2017-09-01 CN disclosed
CN-106317056-A Pyrazolopyridine derivatives, preparation process therefor and therapeutic use thereof 赛诺菲 2017-01-11 CN disclosed