Pyrrole

Pyrrole

SCHEMBL28114401

N#Cc1cccnc1C#N.c1cc[nH]c1

nearest known ligand 0.42

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Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 1/20 0.42
CYP11B1 P15538 1/20 0.40
HPGD P15428 6/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
CYP2C9 P11712 2/20 0.39
CYP2C19 P33261 2/20 0.39
CYP3A4 P08684 1/20 0.39
ALDH1A1 P00352 6/20 0.37
KDM4E B2RXH2 1/20 0.37
DRD2 P14416 1/20 0.37
HTR2A P28223 1/20 0.37
MCL1 Q07820 1/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
POLB P06746 1/20 0.36
PLCG1 P19174 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.35
NPSR1 Q6W5P4 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18611 0.88 LRRK2 (0.46) LRRK2CYP11B1HPGDCYP1A2CYP2D6
SCHEMBL29533314 0.88 LRRK2 (0.46) LRRK2CYP11B1HPGDCYP1A2CYP2D6
SCHEMBL30320148 0.75 PLCG1 (0.41) LRRK2CYP11B1HPGDCYP1A2CYP2D6
SCHEMBL12754871 0.75 GRM5 (0.46) LRRK2CYP11B1HPGDCYP1A2CYP2D6
SCHEMBL167824 0.75 PLCG1 (0.41) LRRK2CYP11B1HPGDCYP1A2CYP2D6
SCHEMBL972357 0.75 LRRK2 (0.42) LRRK2CYP11B1HPGDCYP1A2CYP2D6
SCHEMBL3248902 0.75 PLCG1 (0.41) LRRK2CYP11B1HPGDCYP1A2CYP2D6
Cyclohexane SCHEMBL507539 0.70 GRM5 (0.43) LRRK2HPGDCYP1A2CYP2D6CYP2C9
SCHEMBL29489584 0.70
SCHEMBL155110 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104066730-B Heterocyclic compounds and their use as type III receptor tyrosine kinase modulators 埃姆比特生物科学公司 2017-03-08 CN disclosed