SCHEMBL28124169

SCHEMBL28124169

Nc1cccnc1C(=O)S

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 3/20 0.47
KDM4E B2RXH2 3/20 0.45
MAPT P10636 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
ALDH1A1 P00352 1/20 0.45
CYP3A4 P08684 1/20 0.45
ALOX15 P16050 1/20 0.45
TSHR P16473 1/20 0.45
BLM P54132 1/20 0.45
AGER Q15109 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
NAPRT Q6XQN6 1/20 0.44
PIM1 P11309 1/20 0.43
PIM3 Q86V86 1/20 0.43
TLR7 Q9NYK1 1/20 0.43
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20558075 0.84 GRM4 (0.49) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL128343 0.83 KDM4E (0.61) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL29385675 0.83 MKNK1 (0.49) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL699068 0.83 MKNK1 (0.49) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL29262306 0.81 KDM4E (0.59) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL3380838 0.81 GRM4 (0.46) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL2280224 0.81 KDM4E (0.59) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL4172344 0.79 GRM4 (0.45) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL2280222 0.79 GRM4 (0.45) GRM4KDM4EMAPTL3MBTL1ALDH1A1
SCHEMBL18187340 0.79 GRM4 (0.45) GRM4KDM4EMAPTL3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103946223-B 3-cyanaryl-1h-pyrazolo[2.3-b]pyridine derivatives 默克专利股份公司 2017-01-18 CN disclosed