Cystamine

Cystamine

SCHEMBL28125490

CC(=O)O.N=C(N)N.NCCSSCCN

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Cystamine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 known ✓ P29475 5/20 0.42
NOS2 known ✓ P35228 6/20 0.32
NOS3 known ✓ P29474 4/20 0.32
TSHR P16473 3/20 0.48
THPO P40225 1/20 0.48
MAPT P10636 4/20 0.46
TDP1 Q9NUW8 3/20 0.46
EHMT2 Q96KQ7 1/20 0.46
CYP2C19 P33261 3/20 0.42
CYP1A2 P05177 2/20 0.42
LMNA P02545 2/20 0.41
CYP3A4 P08684 1/20 0.41
APEX1 P27695 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
FFAR3 O14843 1/20 0.33
LCK P06239 1/20 0.33
FYN P06241 1/20 0.33
IDO1 P14902 1/20 0.32
ALOX15 P16050 1/20 0.32
BLM P54132 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Cystamine SCHEMBL9187228 0.90 TSHR (0.59) TSHRTHPOMAPTTDP1EHMT2
Cystamine SCHEMBL445194 0.82 TSHR (0.62) TSHRTHPOMAPTTDP1EHMT2
Cystamine SCHEMBL31646100 0.82 TSHR (0.62) TSHRTHPOMAPTTDP1EHMT2
Acetic Acid SCHEMBL28203493 0.82 FFAR3 (0.44) TSHRMAPTTDP1NOS1CYP2C19
Cystamine SCHEMBL9417963 0.79 TSHR (0.67) TSHRTHPOMAPTTDP1EHMT2
Benzene SCHEMBL28038565 0.77 FFAR3 (0.39) TSHRCYP2C19CYP1A2LMNASMN1; SMN2
Acetic Acid SCHEMBL28261678 0.77 TSHR (0.44) TSHRMAPTTDP1NOS1CYP2C19
Cystamine SCHEMBL28174375 0.77 TSHR (0.56) TSHRTHPOMAPTTDP1EHMT2
Cystamine SCHEMBL2693177 0.76 TDP1 (0.57) TSHRTHPOMAPTTDP1EHMT2
Acetic Acid SCHEMBL8850911 0.76 FFAR3 (0.58) TSHRTHPOMAPTTDP1NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104673096-B Method for preparing coating with nitric oxide (NO) catalytic activity 西南交通大学 2017-05-17 CN claimed