SCHEMBL28146282

SCHEMBL28146282

O=C(Nc1ccc(N(CCCl)CCCl)cc1)c1ccccc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.68
ERBB2 P04626 3/20 0.68
PTPN1 P18031 2/20 0.57
SMO Q99835 1/20 0.56
NPC1 O15118 4/20 0.56
RAB9A P51151 4/20 0.56
MEN1 O00255 2/20 0.56
KMT2A Q03164 2/20 0.56
SIRT1 Q96EB6 1/20 0.56
KDM4E B2RXH2 1/20 0.56
POLB P06746 1/20 0.56
MAPT P10636 1/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
CACNA1B Q00975 1/20 0.53
APBA1 Q02410 1/20 0.53
HDAC1 Q13547 1/20 0.52
HDAC2 Q92769 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
PRMT1 Q99873 1/20 0.51
FFAR1 O14842 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28232821 0.86 EGFR (0.71) EGFRERBB2NPC1RAB9AMEN1
SCHEMBL31060864 0.85 EGFR (0.73) EGFRERBB2NPC1RAB9AMEN1
SCHEMBL15097414 0.84 KMT2A (0.66) EGFRERBB2NPC1RAB9AMEN1
SCHEMBL28468321 0.84 EGFR (0.65) EGFRERBB2HDAC1HDAC2HDAC6
SCHEMBL9122523 0.82 HDAC6 (0.59) EGFRERBB2NPC1RAB9AMEN1
SCHEMBL28477425 0.81 EGFR (0.60) EGFRERBB2PTPN1SMOMEN1
SCHEMBL126415 0.79 PTPN1 (0.87) PTPN1SMONPC1RAB9AMEN1
SCHEMBL28469673 0.79 EGFR (0.69) EGFRERBB2HDAC1HDAC2HDAC6
SCHEMBL29212211 0.78 PTPN1 (0.67) PTPN1SMONPC1RAB9AMEN1
SCHEMBL4910692 0.78 HDAC6 (0.59) EGFRERBB2NPC1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106631856-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-benzoyl -1,4- phenylenediamine and preparation method thereof 长安大学 2019-03-19 CN claimed
CN-106631856-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-benzoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN claimed
CN-106631856-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-benzoyl -1,4- phenylenediamine and preparation method thereof 长安大学 2019-03-19 CN disclosed
CN-106631856-B Nitrogen mustard derivatives N, N- bis- (2- chloroethyl)-N '-benzoyl -1,4- phenylenediamine and preparation method thereof 长安大学 2019-03-19 CN disclosed
CN-106631856-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-benzoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
CN-106631856-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-benzoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed
CN-106631856-A Nitrogen mustard derivative N,N-di(2-chloroethyl)-N'-benzoyl-1,4-phenylenediamine and preparation method thereof 长安大学 2017-05-10 CN disclosed