SCHEMBL28148124

SCHEMBL28148124

O=C(NC1CC1)c1ccc2cnccc2c1

nearest known ligand 0.87

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SMYD3 Q9H7B4 3/20 0.87
MAPK14 Q16539 2/20 0.65
LCK P06239 1/20 0.65
CSF1R P07333 1/20 0.65
KDR P35968 1/20 0.65
HPGDS O60760 2/20 0.56
DRD4 P21917 1/20 0.55
PRMT3 O60678 2/20 0.54
CYP46A1 Q9Y6A2 1/20 0.53
AKT1 P31749 4/20 0.53
CDK2 P24941 1/20 0.52
CYP17A1 P05093 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19710016 0.93 SMYD3 (1.00) SMYD3MAPK14LCKCSF1RKDR
SCHEMBL21490065 0.93 SMYD3 (1.00) SMYD3MAPK14LCKCSF1RKDR
SCHEMBL19710464 0.88 SMYD3 (1.00) SMYD3MAPK14LCKCSF1RKDR
SCHEMBL21490103 0.88 SMYD3 (1.00) SMYD3MAPK14LCKCSF1RKDR
SCHEMBL28437816 0.80 SMYD3 (0.58) SMYD3AKT1CDK2
SCHEMBL28975684 0.80 DRD4 (0.67) SMYD3DRD4
SCHEMBL518025 0.79 SMYD3 (0.63) SMYD3HPGDS
SCHEMBL26928554 0.79 SMYD3 (0.58) SMYD3MAPK14PRMT3AKT1CDK2
SCHEMBL1519811 0.78 SMYD3 (0.60) SMYD3AKT1CDK2
SCHEMBL17643849 0.78 SMYD3 (0.57) SMYD3HPGDSPRMT3AKT1CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106817900-A Novel naphthyridines and isoquinolin and its purposes as CDK8/19 inhibitor 默克专利有限公司 2017-06-09 CN disclosed