SCHEMBL28159092

SCHEMBL28159092

FC(F)(F)c1cccc(Nc2ncnc3ccc(I)cc23)c1

nearest known ligand 0.76

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
EGFR P00533 13/20 0.76
ABCG2 Q9UNQ0 2/20 0.73
TSHR P16473 1/20 0.71
HTT P42858 1/20 0.71
CD38 P28907 1/20 0.67
BRAF P15056 1/20 0.60
CA2 P00918 1/20 0.56
CA9 Q16790 1/20 0.56
AURKB Q96GD4 1/20 0.53
KDR P35968 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3001623 0.86 EGFR (1.00) EGFRABCG2TSHRHTTCD38
SCHEMBL5740246 0.86 CNR1 (0.62) EGFRABCG2TSHRHTTCD38
SCHEMBL8373657 0.85 EGFR (0.76) EGFRABCG2TSHRHTTCD38
SCHEMBL30395473 0.83 EGFR (0.71) EGFRABCG2HTTCD38BRAF
SCHEMBL29058751 0.83 EGFR (0.71) EGFRABCG2HTTCD38BRAF
SCHEMBL8644631 0.82 EGFR (0.71) EGFRABCG2TSHRHTTCD38
SCHEMBL3320018 0.82 EGFR (0.58) EGFRABCG2TSHRHTTCD38
SCHEMBL1192879 0.81 EGFR (0.70) EGFRABCG2TSHRHTTCD38
SCHEMBL29971755 0.81 EGFR (0.70) EGFRABCG2TSHRHTTCD38
SCHEMBL18292535 0.81 RAF1 (0.72) EGFRHTTBRAFKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106986895-A Quinazoline ditosylate salt Mutiple Targets antitumoral compounds and its preparation method and application 北京大学 2017-07-28 CN disclosed