SCHEMBL2816679

SCHEMBL2816679

CC1NC(=N)NC1=O

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6100849 0.72
SCHEMBL21767 0.72
SCHEMBL8110002 0.72
SCHEMBL7240745 0.70
SCHEMBL13074412 0.70 TSHR (0.58)
SCHEMBL16316014 0.70 TSHR (0.58)
SCHEMBL13399686 0.70 TSHR (0.58)
SCHEMBL12809719 0.70 TSHR (0.58)
SCHEMBL1226598 0.70 TSHR (0.58)
SCHEMBL14005348 0.70 TSHR (0.58)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020114530-A1 KIT CONTAINING A BIOLOGICALLY ACTIVE PREPARATION CONTIPRO A.S. (CZ) 2020-06-11 WO claimed
EP-3322488-A1 COSMETIC COMPOSITION Bakel S.R.L. (IT) 2018-05-23 EP claimed
EP-3060195-A1 COSMETIC COMPOSITION BASED ON HYALURONIC ACID, METHOD OF PREPARATION AND USE THEREOF Contipro Biotech s.r.o. (CZ) 2016-08-31 EP claimed
WO-2015058734-A1 COSMETIC COMPOSITION BASED ON HYALURONIC ACID, METHOD OF PREPARATION AND USE THEREOF CONTIPRO BIOTECH S.R.O. (CZ) 2015-04-30 WO claimed
WO-2009046116-A1 SKIN CARE PRODUCTS CONTAINING MULTIPLE ENHANCERS GROSS DENNIS (US) 2009-04-09 WO claimed
WO-2025088285-A1 ECOBIOLOGICAL TOPICAL COMPOSITION FOR TREATING SKIN REDNESS AND DISCOMFORT NAOS INSTITUTE OF LIFE SCIENCE (FR) 2025-05-01 WO disclosed
US-11964039-B2 Compositions that brighten skin, provide sun protection, and permit vitamin D production ARMSTRONG ERNEST T (US) 2024-04-23 US disclosed
US-20220016010-A1 COMPOSITIONS THAT BRIGHTEN SKIN, PROVIDE SUN PROTECTION, AND PERMIT VITAMIN D PRODUCTION ARMSTRONG ERNEST T (US) 2022-01-20 US disclosed
US-11077044-B2 Compositions that brighten skin, provide sun protection, and permit vitamin D production ARMSTRONG ERNEST T (US) 2021-08-03 US disclosed
WO-2020114530-A1 KIT CONTAINING A BIOLOGICALLY ACTIVE PREPARATION CONTIPRO A.S. (CZ) 2020-06-11 WO disclosed
US-20190076346-A1 COMPOSITIONS THAT BRIGHTEN SKIN, PROVIDE SUN PROTECTION, AND PERMIT VITAMIN D PRODUCTION ARMSTRONG ERNEST T (US) 2019-03-14 US disclosed
EP-3405264-A1 COMPOSITIONS THAT BRIGHTEN SKIN, PROVIDE SUN PROTECTION, AND PERMIT VITAMIN D PRODUCTION Armstrong, Ernest T. (AU) 2018-11-28 EP disclosed
EP-3322488-A1 COSMETIC COMPOSITION Bakel S.R.L. (IT) 2018-05-23 EP disclosed
WO-2017124156-A1 COMPOSITIONS THAT BRIGHTEN SKIN, PROVIDE SUN PROTECTION, AND PERMIT VITAMIN D PRODUCTION ARMSTRONG ERNEST T (AU) 2017-07-27 WO disclosed
EP-3060195-A1 COSMETIC COMPOSITION BASED ON HYALURONIC ACID, METHOD OF PREPARATION AND USE THEREOF Contipro Biotech s.r.o. (CZ) 2016-08-31 EP disclosed
WO-2015058734-A1 COSMETIC COMPOSITION BASED ON HYALURONIC ACID, METHOD OF PREPARATION AND USE THEREOF CONTIPRO BIOTECH S.R.O. (CZ) 2015-04-30 WO disclosed
US-20100247476-A1 Copolymer Containing Water-Soluble Lipids Societe d'Exploitation de Products Pour Les Industries Chimiques SEPPIC (FR) 2010-09-30 US disclosed
WO-2009046116-A1 SKIN CARE PRODUCTS CONTAINING MULTIPLE ENHANCERS GROSS DENNIS (US) 2009-04-09 WO disclosed