SCHEMBL28189031

SCHEMBL28189031

Nc1cccc(C=Cc2ccc(O)c(-c3ccccn3)c2)c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 17/20 1.00
CYP19A1 P11511 2/20 0.49
MAOA P21397 1/20 0.49
MAOB P27338 1/20 0.49
NPC1 O15118 1/20 0.48
MAPT P10636 1/20 0.48
GFER P55789 1/20 0.48
HDAC1 Q13547 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC6 Q9UBN7 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28189029 1.00 KDM1A (1.00) KDM1ACYP19A1MAOAMAOBNPC1
SCHEMBL4919409 0.81 KDM1A (0.70) KDM1ANPC1MAPT
SCHEMBL6797387 0.75 CYP19A1 (0.63) KDM1ACYP19A1MAOAMAOBNPC1
SCHEMBL6797384 0.75 CYP19A1 (0.63) KDM1ACYP19A1MAOAMAOBNPC1
SCHEMBL5687683 0.73 KDM1A (0.59) KDM1ANPC1MAPT
Hydrochloric Acid SCHEMBL5687735 0.71 KDM1A (0.57) KDM1ANPC1MAPT
SCHEMBL11288404 0.70 CYP19A1 (0.91) KDM1ACYP19A1MAOAMAOBNPC1
SCHEMBL11288405 0.70 CYP19A1 (0.91) KDM1ACYP19A1MAOAMAOBNPC1
SCHEMBL2774532 0.70 CYP19A1 (0.86) KDM1ACYP19A1MAOAMAOBNPC1
SCHEMBL29664559 0.70 CYP19A1 (0.86) KDM1ACYP19A1MAOAMAOBNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107501169-A A kind of trans diarylethene LSD1 inhibitor, its preparation method and application 新乡医学院 2017-12-22 CN disclosed