SCHEMBL28209587

SCHEMBL28209587

CC(C)(C)OC(=O)Nc1cc(C(=O)O)cnc1CCO

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
BRD9 Q9H8M2 1/20 0.35
MAPT P10636 1/20 0.34
MAPKAPK2 P49137 6/20 0.34
CYP17A1 P05093 2/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
NAMPT P43490 1/20 0.34
METAP1 P53582 1/20 0.34
BRD4 O60885 1/20 0.34
CNR2 P34972 1/20 0.33
GRIN2B Q13224 1/20 0.33
ATR Q13535 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31078088 0.84 AAK1 (0.44) MAPKAPK2GSK3BDYRK1AMETAP1
SCHEMBL29878128 0.80 BRD9 (0.40) BRD9MAPTCYP17A1GSK3BDYRK1A
SCHEMBL5489930 0.80 BRD9 (0.40) BRD9MAPTCYP17A1GSK3BDYRK1A
SCHEMBL18940478 0.80 ATR (0.41) MAPKAPK2CYP17A1GSK3BDYRK1ANAMPT
SCHEMBL18961365 0.80 CYP17A1 (0.38) BRD9MAPKAPK2CYP17A1GSK3BDYRK1A
SCHEMBL14822488 0.74 ATR (0.40) MAPTMAPKAPK2ATR
SCHEMBL2258337 0.72 MAPT (0.42) MAPTMAPKAPK2CYP17A1NAMPTGRIN2B
SCHEMBL15862073 0.72 NAMPT (0.39) MAPTMAPKAPK2DYRK1ANAMPT
SCHEMBL31439890 0.71 GSK3B (0.39) BRD9MAPKAPK2CYP17A1GSK3BDYRK1A
SCHEMBL3256083 0.71 NPC1 (0.54) BRD9MAPTCYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107922386-A 1,4 disubstituted imidazolium derivatives 大日本住友制药株式会社 2018-04-17 CN disclosed
CN-107922348-A Bicyclic heterocyclic amide derivatives 大日本住友制药株式会社 2018-04-17 CN disclosed