SCHEMBL28211527

SCHEMBL28211527

O=CC1(Br)CCCN1c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.36
OPRL1 P41146 1/20 0.36
SLC6A9 P48067 1/20 0.36
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
ALOX12 P18054 1/20 0.35
CYP3A4 P08684 4/20 0.34
CYP2C19 P33261 3/20 0.34
USP2 O75604 2/20 0.34
ALDH1A1 P00352 2/20 0.34
CYP2D6 P10635 1/20 0.34
TSHR P16473 1/20 0.34
HIF1A Q16665 2/20 0.33
FFAR1 O14842 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
HSD17B10 Q99714 1/20 0.33
CYP1A2 P05177 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836402 0.72 CYP3A4 (0.39) OPRM1OPRL1SLC6A9GAACYP3A4
SCHEMBL27777593 0.70 GRIN2D (0.41) OPRM1OPRL1SLC6A9LMNAGAA
SCHEMBL8452213 0.68 USP2 (0.39) OPRM1OPRL1SLC6A9LMNACYP3A4
SCHEMBL22455050 0.68 AR (0.47) OPRM1OPRL1SLC6A9LMNACYP3A4
SCHEMBL28286498 0.68 USP2 (0.39) OPRM1OPRL1SLC6A9LMNACYP3A4
SCHEMBL2899064 0.67 CYP3A4 (0.40) OPRM1OPRL1SLC6A9CYP3A4CYP2C19
SCHEMBL28193878 0.66 FFAR1 (0.38) OPRM1OPRL1SLC6A9LMNACYP3A4
SCHEMBL15059997 0.66 FFAR1 (0.44) CYP3A4CYP2C19USP2ALDH1A1CYP2D6
SCHEMBL2733709 0.64 NR1H2 (0.52) OPRM1OPRL1SLC6A9LMNACYP3A4
SCHEMBL2733711 0.64 NR1H2 (0.52) OPRM1OPRL1SLC6A9LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107849044-A Thriazaspiro last of the ten Heavenly stems ketone compounds as DDR1 inhibitor 豪夫迈·罗氏有限公司 2018-03-27 CN disclosed