SCHEMBL28215216

SCHEMBL28215216

CCc1cccc(-c2cnc3cc[nH]c3c2)c1

nearest known ligand 0.48

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.48
PIK3C3 Q8NEB9 1/20 0.47
CDK8 P49336 3/20 0.46
BRD4 O60885 1/20 0.46
GRIN2B Q13224 10/20 0.45
FGFR1 P11362 1/20 0.42
NISCH Q9Y2I1 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23600955 0.81 BRD4 (0.52) IDO1PIK3C3BRD4GRIN2B
SCHEMBL28215219 0.79 PIK3C3 (0.48) IDO1PIK3C3BRD4GRIN2B
SCHEMBL4400758 0.78 BRD4 (0.44) IDO1PIK3C3BRD4FGFR1
SCHEMBL18363124 0.78 AXL (0.54) PIK3C3CDK8BRD4
SCHEMBL24721353 0.77 CDK8 (0.50) PIK3C3CDK8BRD4GRIN2B
SCHEMBL28214614 0.74 CDK8 (0.47) PIK3C3CDK8BRD4GRIN2B
SCHEMBL10269696 0.73 NPC1 (0.62) IDO1CDK8BRD4FGFR1
SCHEMBL5547358 0.72 BCL2 (0.62) IDO1FGFR1NISCH
SCHEMBL29489424 0.72 BCL2 (0.62) IDO1FGFR1NISCH
SCHEMBL22878658 0.71 PIK3C3 (0.44) PIK3C3CDK8BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108026094-A Substituted 4-azaindoles and their use as modulators of the G L UN2B receptor 詹森药业有限公司 2018-05-11 CN claimed
CN-108026094-A Substituted 4-azaindoles and their use as modulators of the G L UN2B receptor 詹森药业有限公司 2018-05-11 CN disclosed