SCHEMBL28217150

SCHEMBL28217150

O=C(c1ccc(-c2cccc3ccoc23)cc1)N1CCOCC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 5/20 0.50
JAK2 O60674 2/20 0.50
JAK1 P23458 2/20 0.50
TYK2 P29597 2/20 0.50
JAK3 P52333 2/20 0.50
PHGDH O43175 1/20 0.49
HDAC4 P56524 1/20 0.48
RIPK1 Q13546 1/20 0.47
ERN1 O75460 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
ALDH1A1 P00352 1/20 0.47
TSHR P16473 1/20 0.47
MEN1 O00255 1/20 0.46
RAB9A P51151 1/20 0.46
KMT2A Q03164 1/20 0.46
MAPK10 P53779 1/20 0.46
PDCD1 Q15116 1/20 0.46
CD274 Q9NZQ7 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21316005 0.77 JAK2 (0.48) HPGDJAK2JAK1TYK2JAK3
SCHEMBL16345943 0.77 HRH3 (0.48) HPGDJAK2JAK1TYK2JAK3
SCHEMBL16345139 0.77 PDCD1 (0.49) HPGDJAK2JAK1TYK2JAK3
SCHEMBL8150805 0.76 HPGD (0.76) HPGDPHGDHALDH1A1TSHRMEN1
SCHEMBL31622701 0.76 PHGDH (0.53) HPGDJAK2PHGDHHDAC4ERN1
SCHEMBL13952297 0.75 HPGD (0.60) HPGDPHGDHHDAC4RIPK1ERN1
SCHEMBL10720943 0.74 PHGDH (0.81) HPGDPHGDHALDH1A1TSHRKMT2A
SCHEMBL31622597 0.74 ERN1 (0.49) HPGDJAK2PHGDHHDAC4ERN1
SCHEMBL31622683 0.73 ERN1 (0.61) HPGDJAK2PHGDHHDAC4ERN1
SCHEMBL26184965 0.72 MAPT (0.38) HPGDCYP1A2CYP3A4ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108440515-A Substituted benzofuranyl and benzoxazole based compound and application thereof 卡尔约药物治疗公司 2018-08-24 CN disclosed
CN-105492437-B Substituted benzofuranyl and benzoxazolyl compounds and uses thereof 卡尔约药物治疗公司 2018-05-11 CN disclosed