SCHEMBL28218318

SCHEMBL28218318

Fc1ccc2c3c([nH]c2c1)C(C(F)(F)F)=Nc1ccccc1C3

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 9/20 0.49
CA2 P00918 9/20 0.49
CA4 P22748 9/20 0.49
CA6 P23280 9/20 0.49
PARP1 P09874 2/20 0.41
CCNB2 O95067 2/20 0.37
CDK1 P06493 2/20 0.37
CCNB1 P14635 2/20 0.37
GSK3B P49841 2/20 0.37
CDK5 Q00535 2/20 0.37
CDK5R1 Q15078 2/20 0.37
CCNB3 Q8WWL7 2/20 0.37
GSK3A P49840 1/20 0.37
MAPK10 P53779 2/20 0.36
RIPK1 Q13546 2/20 0.36
ACHE P22303 2/20 0.36
BCHE P06276 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
KCNH2 Q12809 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28217847 0.88 CA1 (0.47) CA1CA2CA4CA6CCNB2
SCHEMBL28218315 0.81 GSK3B (0.44) CA1CA2CA4CA6CCNB2
SCHEMBL28217857 0.81 CDK1 (0.52) CA1CA2CA4CA6CCNB2
SCHEMBL28217889 0.77 CCNB2 (0.43) CA1CA2CA4CA6CCNB2
SCHEMBL2299152 0.76 CA1 (0.71) CA1CA2CA4CA6PARP1
SCHEMBL28218316 0.75 CFTR (0.34) CA1CA2CA4CA6PARP1
SCHEMBL2296063 0.66 CA1 (0.83) CA1CA2CA4CA6PARP1
SCHEMBL8946292 0.65 CA1 (0.71) CA1CA2CA4CA6PARP1
SCHEMBL12382617 0.62 CA1 (0.58) CA1CA2CA4CA6PARP1
SCHEMBL29562978 0.62 AHR (0.64) CA1CA2CA4CA6CCNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108101912-A Dihydrobenzene nitrogen Zhuo diindyl derivative and preparation method thereof 浙江大学 2018-06-01 CN disclosed