SCHEMBL28218792

SCHEMBL28218792

COC(=O)c1cccc(CNc2ccc(C)cc2)c1

nearest known ligand 0.72

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 3/20 0.72
CA1 P00915 2/20 0.62
CA2 P00918 2/20 0.62
SENP1 Q9P0U3 2/20 0.62
LOXL2 Q9Y4K0 1/20 0.57
CYP4F2 P78329 2/20 0.56
CYP4A11 Q02928 2/20 0.56
MAPT P10636 2/20 0.53
POLB P06746 1/20 0.53
GAA P10253 1/20 0.53
HTT P42858 1/20 0.53
HDAC8 Q9BY41 1/20 0.52
HDAC6 Q9UBN7 1/20 0.52
EGFR P00533 1/20 0.52
FFAR1 O14842 1/20 0.52
TCF4 P15884 1/20 0.51
CTNNB1 P35222 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15761753 0.88 HIF1A (0.85) HIF1ACA1CA2SENP1LOXL2
SCHEMBL15761744 0.87 HIF1A (0.67) HIF1ACA1CA2SENP1LOXL2
SCHEMBL15755382 0.87 HIF1A (0.70) HIF1ACA1CA2SENP1LOXL2
SCHEMBL15761718 0.87 HIF1A (0.70) HIF1ACA1CA2SENP1LOXL2
SCHEMBL16550428 0.85 HIF1A (0.70) HIF1AHTTHDAC8HDAC6FFAR1
SCHEMBL18300943 0.83 HIF1A (0.61) HIF1ACA1CA2SENP1LOXL2
SCHEMBL17618029 0.82 CA1 (0.77) CA1CA2LOXL2MAPTPOLB
SCHEMBL15761745 0.81 HIF1A (0.65) HIF1ACA1CA2SENP1LOXL2
SCHEMBL15761730 0.81 HIF1A (0.65) HIF1ACA1CA2SENP1LOXL2
SCHEMBL15761741 0.81 HIF1A (0.65) HIF1ACA1CA2SENP1LOXL2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137518-A As 6 inhibitor of histone deacetylase 1,3,4- oxadiazole derivatives compound and include its pharmaceutical composition 株式会社钟根堂 2018-06-08 CN disclosed