SCHEMBL28220075

SCHEMBL28220075

CNC(=O)c1ccc(CC(F)(F)F)cn1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 4/20 0.47
PARP2 Q9UGN5 3/20 0.44
TNKS O95271 2/20 0.44
KCNH2 Q12809 1/20 0.44
ALDH1A1 P00352 2/20 0.42
KDR P35968 2/20 0.42
PIP5K1C O60331 1/20 0.40
PIK3CA P42336 1/20 0.40
PI4KA P42356 1/20 0.40
PI4KB Q9UBF8 1/20 0.40
RAF1 P04049 4/20 0.40
HIF1A Q16665 2/20 0.39
EPAS1 Q99814 1/20 0.39
P4HTM Q9NXG6 1/20 0.39
PARP6 Q2NL67 2/20 0.39
PARP3 Q9Y6F1 2/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1584750 0.81 MAPK1 (0.54) PARP1ALDH1A1HIF1AP4HTMKDM4E
SCHEMBL1584427 0.80 P4HTM (0.61) ALDH1A1HIF1AP4HTMKDM4EMEN1
SCHEMBL30027907 0.80 PARP1 (0.51) PARP1ALDH1A1PIP5K1CPIK3CAPI4KA
SCHEMBL26970993 0.80 PARP1 (0.51) PARP1ALDH1A1PIP5K1CPIK3CAPI4KA
SCHEMBL16597438 0.80 PARP1 (0.51) PARP1ALDH1A1PIP5K1CPIK3CAPI4KA
SCHEMBL12561176 0.80 PLK1 (0.55) PARP1PARP2KCNH2ALDH1A1PIP5K1C
SCHEMBL2642500 0.79 PARP1 (0.50) PARP1ALDH1A1KDRPIP5K1CPIK3CA
SCHEMBL2642502 0.79 PARP1 (0.50) PARP1ALDH1A1PIP5K1CPIK3CAPI4KA
SCHEMBL26970992 0.79 PARP1 (0.50) PARP1ALDH1A1PIP5K1CPIK3CAPI4KA
SCHEMBL17091441 0.78 PARP1 (0.47) PARP1ALDH1A1HIF1AP4HTMKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108137513-A Pyrimidine derivatives ASKA 制药株式会社 2018-06-08 CN disclosed