SCHEMBL28223904

SCHEMBL28223904

O=C1NCc2c1cccc2-c1ccc(F)cc1

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.64
PIK3CA P42336 1/20 0.64
PIK3CB P42338 1/20 0.64
GRM2 Q14416 1/20 0.63
KDR P35968 12/20 0.60
CLK4 Q9HAZ1 4/20 0.54
PIM1 P11309 4/20 0.54
ROCK1 Q13464 4/20 0.54
DYRK1A Q13627 3/20 0.54
CDK5 Q00535 2/20 0.54
CSNK1A1 P48729 1/20 0.54
LRRK2 Q5S007 1/20 0.54
DYRK1B Q9Y463 1/20 0.54
LTK P29376 1/20 0.51
MST1R Q04912 1/20 0.51
ROCK2 O75116 4/20 0.50
MAP4K4 O95819 3/20 0.50
STK3 Q13188 3/20 0.50
NTRK3 Q16288 3/20 0.50
TAOK1 Q7L7X3 3/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1335607 0.86 KDR (0.82) KDRCLK4PIM1ROCK1ROCK2
SCHEMBL30331758 0.84 PARP10 (0.69) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL1333209 0.83 KDR (0.57) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL19608227 0.83 PIK3CD (0.64) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL29845432 0.81 CLK4 (0.57) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL30775282 0.80 KDR (0.58) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL30775285 0.79 KDR (0.57) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL28860691 0.79 KDR (0.54) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL30543353 0.79 KDR (0.62) PIK3CDPIK3CAPIK3CBKDRCLK4
SCHEMBL1333899 0.79 KDR (0.65) KDRCLK4PIM1ROCK1DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368053-A Substituted benzazepine derivatives as antibacterial compounds 葛兰素史密斯克莱知识产权发展有限公司 2018-08-03 CN disclosed