SCHEMBL28223905

SCHEMBL28223905

O=C1NCc2c1cccc2-c1ccccc1F

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 3/20 0.56
CDK5 Q00535 2/20 0.56
DYRK1A Q13627 2/20 0.56
ROCK1 Q13464 2/20 0.56
PIM1 P11309 1/20 0.56
CSNK1A1 P48729 1/20 0.56
LRRK2 Q5S007 1/20 0.56
DYRK1B Q9Y463 1/20 0.56
PIK3CD O00329 2/20 0.54
PIK3CB P42338 2/20 0.54
PIK3CA P42336 1/20 0.54
LTK P29376 1/20 0.53
MST1R Q04912 1/20 0.53
KDR P35968 8/20 0.51
CA12 O43570 1/20 0.48
CA9 Q16790 1/20 0.48
GRM2 Q14416 1/20 0.45
PARP10 Q53GL7 1/20 0.44
PARP11 Q9NR21 1/20 0.44
PARP1 P09874 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29871952 0.87 CDK5 (0.61) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL1078443 0.87 CDK5 (0.61) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30775381 0.82 CLK4 (0.49) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL1334382 0.81 KDR (0.54) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30543362 0.79 KDR (0.49) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30775229 0.79 PARP1 (0.57) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30775244 0.79 PARP10 (0.57) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30775289 0.78 KDR (0.54) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30775251 0.78 CLK4 (0.51) CLK4CDK5DYRK1AROCK1PIM1
SCHEMBL30331758 0.78 PARP10 (0.69) CLK4CDK5DYRK1AROCK1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108368053-A Substituted benzazepine derivatives as antibacterial compounds 葛兰素史密斯克莱知识产权发展有限公司 2018-08-03 CN disclosed