SCHEMBL28239774

SCHEMBL28239774

[CH2]C1(C)CNc2ccccc21

nearest known ligand 0.39

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 1/20 0.39
PDK4 Q16654 1/20 0.39
KDM1A O60341 1/20 0.37
HTR5A P47898 4/20 0.36
ATM Q13315 1/20 0.35
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
BRD4 O60885 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRL1 P41146 1/20 0.33
BACE1 P56817 1/20 0.33
ALOX15 P16050 1/20 0.32
HSD17B10 Q99714 1/20 0.32
POLB P06746 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29384370 0.78 PDK2 (0.42) PDK2PDK4KDM1AHTR5AATM
SCHEMBL1031209 0.78 PDK2 (0.42) PDK2PDK4KDM1AHTR5AATM
Hydrochloric Acid SCHEMBL2482151 0.77 PDK2 (0.41) PDK2PDK4KDM1AHTR5AATM
SCHEMBL24124146 0.75 PDK2 (0.39) PDK2PDK4KDM1AHTR5AATM
SCHEMBL2349269 0.75 PDK2 (0.39) PDK2PDK4KDM1AHTR5AATM
SCHEMBL27491877 0.73 KDM1A (0.40) PDK2PDK4KDM1AHTR5AATM
SCHEMBL26295503 0.72 PDK2 (0.37) PDK2PDK4KDM1AHTR5AATM
SCHEMBL16566109 0.72 KDM1A (0.39) PDK2PDK4KDM1AHTR5AATM
SCHEMBL20506223 0.71 BRD4 (0.37) PDK2PDK4KDM1AHTR5AATM
SCHEMBL1094251 0.71 PDK2 (0.40) PDK2PDK4KDM1AHTR5AATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108495855-A Condesned thiazole and pyrimidine derivatives as MNK inhibitor 生命弧度公司 2018-09-04 CN disclosed