SCHEMBL28243649

SCHEMBL28243649

COc1ccc2c(-c3ccnc(Nc4cc(N)c(N(C)CCN(C)C)cc4OC)n3)cn(C(F)F)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 19/20 0.53
MKNK1 Q9BUB5 1/20 0.52
MKNK2 Q9HBH9 1/20 0.52
MLNR O43193 1/20 0.51
KDM1A O60341 1/20 0.51
ABCB11 O95342 1/20 0.51
ERBB2 P04626 1/20 0.51
INSR P06213 1/20 0.51
CHRM2 P08172 1/20 0.51
HTR1A P08908 1/20 0.51
ADORA3 P0DMS8 1/20 0.51
DRD2 P14416 1/20 0.51
NQO2 P16083 1/20 0.51
ADRA2C P18825 1/20 0.51
DRD1 P21728 1/20 0.51
ERBB3 P21860 1/20 0.51
SLC6A2 P23975 1/20 0.51
HTR2A P28223 1/20 0.51
HTR2C P28335 1/20 0.51
ADORA2A P29274 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17553699 0.91 EGFR (0.60) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL28244311 0.88 EGFR (0.52) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL17683081 0.87 EGFR (0.55) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL30459704 0.87 EGFR (0.55) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL28864311 0.85 EGFR (0.72) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL17542611 0.84 MKNK1 (0.65) EGFRMKNK1MKNK2MLNRKDM1A
SCHEMBL19337061 0.82 EGFR (0.64) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL22994937 0.82 EGFR (0.62) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL14660679 0.81 EGFR (0.73) EGFRMLNRKDM1AABCB11ERBB2
SCHEMBL29524806 0.81 EGFR (0.73) EGFRMLNRKDM1AABCB11ERBB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108530428-A Substituted pyrimidine derivatives and preparation method thereof and medicinal usage 四川海思科制药有限公司 2018-09-14 CN disclosed