SCHEMBL28255706

SCHEMBL28255706

O=C1CCC(c2cc(F)ccc2F)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 3/20 0.46
KDM1A O60341 2/20 0.46
KDM1B Q8NB78 1/20 0.46
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
PTGDR2 Q9Y5Y4 2/20 0.40
ESR2 Q92731 1/20 0.39
AKR1A1 P14550 1/20 0.39
AKR1B1 P15121 1/20 0.39
SLC6A2 P23975 2/20 0.37
SLC6A4 P31645 2/20 0.37
SLC6A3 Q01959 2/20 0.37
HTR1A P08908 1/20 0.37
HCRTR2 O43614 1/20 0.37
CHRNB2 P17787 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
HTR2A P28223 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4543678 0.85 OPRL1 (0.46) ESR2AKR1A1AKR1B1HTR2AHTR2C
SCHEMBL15566855 0.84 KDM1A (0.55) HCAR2KDM1AKDM1BPTGDR2AKR1A1
SCHEMBL11830644 0.82 PTGDR2 (0.38) PTGDR2ESR2SLC6A2SLC6A4SLC6A3
SCHEMBL18938470 0.81 KDM1A (0.46) HCAR2KDM1AKDM1BKMT2AMEN1
SCHEMBL426443 0.81 KDM1A (0.53) HCAR2KDM1AKDM1BKMT2AMEN1
SCHEMBL28247579 0.80 KDM1A (0.52) HCAR2KDM1AKDM1BKMT2AMEN1
SCHEMBL11773147 0.80 KDM1A (0.52) HCAR2KDM1AKDM1BKMT2AMEN1
SCHEMBL505573 0.79 OPRL1 (0.48) SLC6A4HTR2AHTR2C
SCHEMBL11830630 0.79 OPRL1 (0.48) PTGDR2ESR2CHRNB2CHRNB4CHRNA3
SCHEMBL1528700 0.79 ESR2 (0.38) ESR2AKR1A1AKR1B1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-114181136-A Substituted piperidine compounds and uses thereof 武田药品工业株式会社 2022-03-15 CN disclosed
CN-108884043-B Substituted piperidine compounds and uses thereof 武田药品工业株式会社 2021-11-26 CN disclosed
CN-108884043-A Substituted piperidine compounds and uses thereof 武田药品工业株式会社 2018-11-23 CN disclosed