SCHEMBL2825824

SCHEMBL2825824

CCn1nc(-c2cccc(Sc3ccc(OC)cc3)c2)cc(N)c1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.38
NTSR1 P30989 1/20 0.37
MAPT P10636 4/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
HDAC1 Q13547 2/20 0.37
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
NPC1 O15118 1/20 0.36
ALDH1A1 P00352 1/20 0.36
STAT1 P42224 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
TGM2 P21980 1/20 0.35
TGM1 P22735 1/20 0.35
CASP3 P42574 1/20 0.35
TGM3 Q08188 1/20 0.35
PTGIR P43119 1/20 0.35
ADORA2A P29274 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2826223 0.93 HDAC1 (0.41) MAPTHDAC1MTNR1AMTNR1BADORA2A
SCHEMBL2826787 0.84 HDAC1 (0.48) MAPTSMN1; SMN2HDAC1MEN1KMT2A
SCHEMBL2825919 0.84 COMT (0.46) MAPTSMN1; SMN2HDAC1MEN1KMT2A
SCHEMBL2826119 0.83 PDE4B (0.39) MAPTHDAC1MEN1KMT2AALDH1A1
SCHEMBL4054330 0.83 MAPT (0.46) MAPTSMN1; SMN2HDAC1MEN1KMT2A
SCHEMBL13291030 0.81 POLB (0.35) MAPTMEN1KMT2AALDH1A1ADORA2A
SCHEMBL2829672 0.80 HDAC1 (0.45) MAPTSMN1; SMN2HDAC1MEN1KMT2A
SCHEMBL2823397 0.76 PDE4B (0.68) ADORA2A
SCHEMBL4061285 0.75 NPC1 (0.47) MAPTSMN1; SMN2KMT2ANPC1ALDH1A1
SCHEMBL2835042 0.75 PDE4B (0.49) ADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010069504-A1 (3-OXO)PYRIDIN-4-YLUREA DERIVATIVES AS PDE4 INHIBITORS ALMIRALL, S.A. (ES) 2010-06-24 WO disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed
EP-2196465-A1 (3-oxo)pyridazin-4-ylurea derivatives as PDE4 inhibitors Almirall, S.A. (ES) 2010-06-16 EP disclosed