SCHEMBL2827083

SCHEMBL2827083

CCCN(CCCO)C(N)=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 5/20 0.41
CA9 Q16790 5/20 0.41
CA2 P00918 3/20 0.41
CA1 P00915 4/20 0.39
TSHR P16473 2/20 0.39
MAPK1 P28482 1/20 0.39
ALDH1A1 P00352 3/20 0.36
HPGD P15428 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP3 P08254 1/20 0.36
MMP8 P22894 1/20 0.36
TP53 P04637 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 2/20 0.33
HSD17B10 Q99714 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NTRK2 Q16620 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2829319 0.91 CA12 (0.48) CA12CA9CA2CA1TSHR
SCHEMBL194060 0.89 NTRK2 (0.36) CA12CA9CA1NTRK2
SCHEMBL2828720 0.86 CA12 (0.44) CA12CA9CA2CA1TSHR
SCHEMBL292931 0.86 CA12 (0.52) CA12CA9CA2CA1TSHR
SCHEMBL107452 0.86 CA12 (0.52) CA12CA9CA2CA1TSHR
SCHEMBL42388 0.86 CA12 (0.52) CA12CA9CA2CA1TSHR
SCHEMBL2829211 0.84 CA12 (0.42) CA12CA9CA2CA1TSHR
SCHEMBL4370605 0.84 CA12 (0.45) CA12CA9CA2CA1TSHR
SCHEMBL2843504 0.84 NTRK2 (0.34) CA12CA9CA2CA1NTRK2
SCHEMBL4058348 0.84 CA12 (0.50) CA12CA9CA2CA1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103635462-A Method for producing acrylic esters BASF SE 2014-03-12 CN disclosed
CN-1993316-B Catalytic methods for the production of (meth)acrylates from n-hydroxyalkylated amides BASF AG 2011-07-20 CN disclosed
EP-1758869-B1 PYRIDAZIN-3(2H)-ONE DERIVATIVES AND THEIR USE AS PDE4 INHIBITORS ALMIRALL SA (ES) 2010-12-22 EP disclosed
US-7511038-B2 Pyridazin-3(2H)-one derivatives and their use as PDE4 inhibitors LABORATORIOS ALMIRALL S.A. (ES) 2009-03-31 US disclosed
EP-1575926-B1 NEW PYRIDAZIN-3(2H)-ONE DERIVATIVES ALMIRALL LAB (ES) 2008-03-05 EP disclosed
CN-1993316-A Catalytic methods for the production of (meth)acrylates from n-hydroxyalkylated amides BASF AG (DE) 2007-07-04 CN disclosed
EP-1781621-A1 PYRIDAZIN-3(2H)-ONE DERIVATIVES AND THEIR USE AS PDE4 INHIBITORS Laboratorios Almirall, S.A. (ES) 2007-05-09 EP disclosed
EP-1682519-A1 PYRIDAZIN-3(2H)-ONE DERIVATIVES AND THEIR USE AS PDE4 INHIBITORS Almirall Prodesfarma, S.A. (ES) 2006-07-26 EP disclosed
WO-2005123693-A1 PYRIDAZIN-3(2H)-ONE DERIVATIVES AND THEIR USE AS PDE4 INHIBITORS LABORATORIOS ALMIRALL, S.A. (ES) 2005-12-29 WO disclosed
EP-1575926-A1 NEW PYRIDAZIN-3(2H)-ONE DERIVATIVES Almirall Prodesfarma, S.A. (ES) 2005-09-21 EP disclosed
WO-2005049581-A1 PYRIDAZIN-3 (2H) -ONE DERIVATIVES AND THEIR USE AS PDE4 INHIBITORS ALMIRALL PRODESFARMA, S.A. (ES) 2005-06-02 WO disclosed
WO-2004058729-A1 NEW PYRIDAZIN-3(2H)-ONE DERIVATIVES ALMIRALL PRODESFARMA SA (ES) 2004-07-15 WO disclosed