SCHEMBL28279239

SCHEMBL28279239

NCc1ccccc1CC(=O)Nc1ccc(-n2cc(Br)cn2)c(S(N)(=O)=O)c1

nearest known ligand 0.47

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
P2RX4 Q99571 18/20 0.47
CA12 O43570 1/20 0.44
CA1 P00915 1/20 0.44
CA2 P00918 1/20 0.44
CA9 Q16790 1/20 0.44
KCNJ6 P48051 1/20 0.43
KCNJ5 P48544 1/20 0.43
KCNJ3 P48549 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19576993 0.93 P2RX4 (0.49) P2RX4CA12CA1CA2CA9
SCHEMBL19551688 0.90 P2RX4 (0.51) P2RX4CA12CA1CA2CA9
SCHEMBL19552060 0.90 P2RX4 (0.59) P2RX4
SCHEMBL19551523 0.90 KCNJ6 (0.51) P2RX4CA12CA1CA2CA9
SCHEMBL28280466 0.89 P2RX4 (0.51) P2RX4
SCHEMBL28870232 0.89 P2RX4 (0.47) P2RX4CA12CA1CA2CA9
SCHEMBL19551595 0.87 P2RX4 (0.53) P2RX4CA12CA1CA2CA9
SCHEMBL28280448 0.87 P2RX4 (0.46) P2RX4CA12CA1CA2CA9
SCHEMBL28280338 0.87 P2RX4 (0.46) P2RX4KCNJ5KCNJ3
SCHEMBL29782414 0.85 P2RX4 (0.47) P2RX4CA12CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109415321-A aromatic sulfonamide derivatives 拜耳制药股份公司 2019-03-01 CN disclosed