SCHEMBL28285702

SCHEMBL28285702

C#Cc1cccc(Nc2nccc(Cl)n2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SYK P43405 2/20 0.47
EGFR P00533 3/20 0.45
GAK O14976 1/20 0.45
EPHB4 P54760 1/20 0.44
AURKA O14965 4/20 0.44
IDO1 P14902 2/20 0.44
TDO2 P48775 2/20 0.44
PRKCD Q05655 2/20 0.43
ABL1 P00519 1/20 0.43
BCR P11274 1/20 0.43
PRKCA P17252 1/20 0.43
CDK2 P24941 3/20 0.43
NPC1 O15118 2/20 0.43
RAB9A P51151 2/20 0.43
AURKB Q96GD4 1/20 0.43
CDK4 P11802 1/20 0.43
FLT3 P36888 1/20 0.43
TYRO3 Q06418 1/20 0.43
MERTK Q12866 1/20 0.43
GAS6 Q14393 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2115684 0.80 ABL1 (0.62) SYKEPHB4PRKCDABL1BCR
SCHEMBL30213680 0.80 ROCK1 (0.49) SYKEGFRGAKEPHB4AURKA
SCHEMBL15522255 0.80 ROCK1 (0.49) SYKEGFRGAKEPHB4AURKA
SCHEMBL22627074 0.80 ABCG2 (0.51) SYKEGFRGAKIDO1TDO2
SCHEMBL30847380 0.78 CDK2 (0.55) SYKEGFREPHB4AURKAPRKCD
SCHEMBL27111928 0.78 CDK2 (0.55) SYKEGFREPHB4AURKAPRKCD
SCHEMBL3439832 0.77 SYK (0.64) SYKAURKAPRKCDABL1BCR
SCHEMBL857880 0.76 AURKA (0.70) EGFREPHB4AURKAPRKCDABL1
SCHEMBL14368039 0.74 CDK5 (0.53) SYKEGFRAURKAIDO1PRKCD
SCHEMBL2113984 0.74 AURKA (0.77) AURKA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109516959-A 2- fragrant amino -4- substituted uracil derivative and its application in preparation of anti-tumor drugs 陕西师范大学 2019-03-26 CN disclosed