SCHEMBL28290827

SCHEMBL28290827

Cc1c(N)cccc1OCCN

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.55
HTR1B P28222 3/20 0.50
TSHR P16473 2/20 0.48
CYP3A4 P08684 1/20 0.48
PIK3CA P42336 1/20 0.48
CYP1A2 P05177 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAPK1 P28482 2/20 0.44
TP53 P04637 1/20 0.44
RAB9A P51151 1/20 0.44
ALDH1A1 P00352 3/20 0.42
HPGD P15428 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
TAAR1 Q96RJ0 1/20 0.41
MAPT P10636 2/20 0.41
GAA P10253 1/20 0.41
TDP1 Q9NUW8 2/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
ADRA2B P18089 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL311482 0.91 HTR1B (0.51) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL21694203 0.85 CYP1A2 (0.61) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL1141672 0.85 CYP1A2 (0.56) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL21694213 0.83 CYP1A2 (0.65) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL21694153 0.83 CYP1A2 (0.65) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL10264421 0.83 CYP1A2 (0.70) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL8489747 0.83 TSHR (0.46) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL10635778 0.83 TSHR (0.46) KDM4EHTR1BTSHRCYP3A4PIK3CA
SCHEMBL7415579 0.82 HTR1B (0.62) KDM4EHTR1BTSHRMAPK1TP53
SCHEMBL23493017 0.81 CYP1A2 (0.62) KDM4EHTR1BTSHRCYP3A4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109563073-A For the treatment of para-5-HT1AReceptor-controlled serotonergic disease-modulating compounds 诺罗利西斯公司 2019-04-02 CN disclosed