SCHEMBL28291947

SCHEMBL28291947

CC(C)(C)c1csc(Nc2ccncc2)n1

nearest known ligand 0.73

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 10/20 0.73
SMN1; SMN2 Q16637 5/20 0.58
TAS1R3 Q7RTX0 1/20 0.58
TAS1R1 Q7RTX1 1/20 0.58
TAS1R2 Q8TE23 1/20 0.58
NPC1 O15118 4/20 0.55
RAB9A P51151 4/20 0.55
MEN1 O00255 2/20 0.55
KMT2A Q03164 2/20 0.55
MAPT P10636 2/20 0.55
TRPV4 Q9HBA0 1/20 0.50
POLB P06746 2/20 0.48
MAPK1 P28482 2/20 0.48
ALDH1A1 P00352 1/20 0.48
VCP P55072 1/20 0.48
ESR1 P03372 1/20 0.48
TDP1 Q9NUW8 1/20 0.48
GAA P10253 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21708025 0.85 CCR4 (0.76) CCR4SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL5486145 0.85 CCR4 (1.00) CCR4SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL21708002 0.82 CCR4 (0.71) CCR4SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL4561810 0.80 CCR4 (0.68) CCR4SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL28297353 0.80 CCR4 (0.68) CCR4SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL12603585 0.77 CCR4 (0.64) CCR4SMN1; SMN2TAS1R3TAS1R1TAS1R2
SCHEMBL21708018 0.76 CCR4 (1.00) CCR4SMN1; SMN2NPC1RAB9AMEN1
SCHEMBL2173513 0.76 CCR4 (0.58) CCR4SMN1; SMN2TAS1R3TAS1R1TAS1R2
SCHEMBL2173118 0.76 CCR4 (0.62) CCR4SMN1; SMN2TAS1R3TAS1R1TAS1R2
SCHEMBL262399 0.76 CCR4 (0.62) CCR4SMN1; SMN2TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106699752-B Application of the 5- piperonyl -2- pridylamino thiazole as anticancer drug 湖南大学 2019-05-14 CN disclosed