SCHEMBL28292658

SCHEMBL28292658

CCc1nc2cc(C)ccc2nc1Br

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NQO2 P16083 1/20 0.50
RAB9A P51151 2/20 0.44
MEN1 O00255 1/20 0.44
NPC1 O15118 1/20 0.44
KMT2A Q03164 1/20 0.44
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
MAPT P10636 4/20 0.42
TDP1 Q9NUW8 1/20 0.42
CYP1A2 P05177 3/20 0.41
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 1/20 0.36
PSMB5 P28074 1/20 0.35
NCK1 P16333 1/20 0.34
BACE1 P56817 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19432353 0.87 NQO2 (0.59) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL10585917 0.82 NQO2 (0.64) NQO2RAB9AKDM4EALDH1A1L3MBTL1
SCHEMBL11421185 0.81 NQO2 (0.53) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL31193100 0.79 KDM4E (0.46) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL30932232 0.77 NQO2 (0.57) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL28286262 0.77 NQO2 (0.57) NQO2RAB9AMEN1KMT2AKDM4E
SCHEMBL19075884 0.77 NQO2 (0.57) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL23280870 0.76 NQO2 (0.47) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL19432431 0.76 NQO2 (0.47) NQO2RAB9AMEN1NPC1KMT2A
SCHEMBL16644141 0.74 NQO2 (0.53) NQO2RAB9AMEN1NPC1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109689647-A The compound that bicyclic heteroaryl replaces 百时美施贵宝公司 2019-04-26 CN disclosed