SCHEMBL28293048

SCHEMBL28293048

Cc1cncc(C#N)c1.O=CCl

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
RAF1 P04049 2/20 0.44
GRM5 P41594 1/20 0.39
CYP11B1 P15538 3/20 0.38
CYP11B2 P19099 3/20 0.38
HCAR2 Q8TDS4 1/20 0.37
P4HTM Q9NXG6 1/20 0.36
ALDH1A1 P00352 1/20 0.35
CYP2A6 P11509 1/20 0.35
SCN10A Q9Y5Y9 2/20 0.35
SCN2A Q99250 1/20 0.35
ATM Q13315 1/20 0.34
KCNH2 Q12809 1/20 0.34
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA3 P32297 1/20 0.33
CHRNA4 P43681 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Formic Acid SCHEMBL28015002 0.91 RAF1 (0.43) RAF1GRM5CYP11B1CYP11B2HCAR2
SCHEMBL29406749 0.90
SCHEMBL149800 0.90
SCHEMBL936524 0.73 CYP11B1 (0.47) RAF1CYP11B1CYP11B2ALDH1A1CHRNB2
SCHEMBL1477361 0.73 GRM5 (0.42) RAF1GRM5SCN10AKCNH2CHRNB2
SCHEMBL1521247 0.73
SCHEMBL3941691 0.72 RAF1 (0.50) RAF1CYP11B1CYP11B2CHRNB2CHRNB4
SCHEMBL31586111 0.72 RAF1 (0.50) RAF1CYP11B1CYP11B2CHRNB2CHRNB4
Formamide SCHEMBL28048213 0.72 CYP11B1 (0.37) RAF1GRM5CYP11B1CYP11B2HCAR2
Formic Acid SCHEMBL27929488 0.72 HCAR2 (0.40) RAF1GRM5CYP11B1CYP11B2HCAR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-106795177-B BACE1 inhibitors 豪夫迈·罗氏有限公司 2019-04-23 CN disclosed