SCHEMBL28293606

SCHEMBL28293606

O=C(c1c(F)ccc(NS(=O)(=O)O)c1F)c1c[nH]c2ncccc12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 5/20 0.63
CYP3A4 P08684 8/20 0.57
CYP2C19 P33261 5/20 0.54
CYP2C9 P11712 5/20 0.54
RIPK2 O43353 2/20 0.54
RAF1 P04049 2/20 0.54
KDR P35968 2/20 0.54
MAP2K2 P36507 2/20 0.54
TGFBR2 P37173 2/20 0.54
NEK2 P51955 2/20 0.54
MAP2K1 Q02750 2/20 0.54
TNK2 Q07912 2/20 0.54
MAP2K5 Q13163 2/20 0.54
PTK6 Q13882 2/20 0.54
NEK11 Q8NG66 2/20 0.54
MAP3K20 Q9NYL2 2/20 0.54
MAP4K5 Q9Y4K4 2/20 0.54
BMPR1B O00238 1/20 0.54
PLK4 O00444 1/20 0.54
PIR O00625 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL298372 0.90 BRAF (0.65) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL298378 0.88 CYP3A4 (0.66) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL855809 0.88 BRAF (0.62) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL297325 0.87 CYP3A4 (0.62) BRAFCYP3A4CYP2C19CYP2C9
SCHEMBL29796856 0.86 BRAF (0.74) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL298039 0.86 BRAF (0.74) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL413713 0.86 BRAF (0.60) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL298432 0.86 CYP3A4 (0.61) BRAFCYP3A4CYP2C19CYP2C9RIPK2
SCHEMBL14620763 0.86 CYP3A4 (0.61) BRAFCYP3A4CYP2C19CYP2C9CYP2D6
SCHEMBL859195 0.85 BRAF (0.69) BRAFCYP3A4CYP2C19CYP2C9CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109608450-A The synthesis of pyrrolo- [2,3-B] pyridine 普莱希科公司 2019-04-12 CN disclosed