SCHEMBL28294330

SCHEMBL28294330

Nc1cc2cn[nH]c2cc1N.[H+]

nearest known ligand 0.95

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.95
KDM4E B2RXH2 2/20 0.55
MEN1 O00255 2/20 0.55
MAPT P10636 2/20 0.55
KMT2A Q03164 2/20 0.55
ROCK2 O75116 2/20 0.55
PKM P14618 1/20 0.55
HTT P42858 1/20 0.55
ALDH1A1 P00352 1/20 0.55
GAA P10253 1/20 0.55
HPGD P15428 1/20 0.55
RAB9A P51151 1/20 0.55
ROCK1 Q13464 1/20 0.55
HIF1A Q16665 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
NOS1 P29475 5/20 0.45
METAP2 P50579 3/20 0.45
DYRK1A Q13627 3/20 0.45
CSNK2A1 P68400 1/20 0.45
MAPK1 P28482 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2268059 0.98 CHEK1 (1.00) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL29589219 0.98 CHEK1 (1.00) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL1273919 0.83 CHEK1 (0.73) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL28642996 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL1273798 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL28858305 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL14389670 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL2568456 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A
SCHEMBL29536144 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A
Hydrochloric Acid SCHEMBL15640013 0.81 CHEK1 (0.70) CHEK1KDM4EMEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109761986-A Three simultaneously ring analog derivative inhibitor, preparation method and applications 上海翰森生物医药科技有限公司 2019-05-17 CN disclosed