SCHEMBL28296355

SCHEMBL28296355

COc1ccc(CNc2ncc3cc(-c4ccccc4Cl)ccc3n2)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CLK4 Q9HAZ1 8/20 0.48
DYRK1A Q13627 3/20 0.48
DYRK1B Q9Y463 3/20 0.48
CLK1 P49759 2/20 0.48
CLK2 P49760 2/20 0.48
RPS6KB1 P23443 2/20 0.48
ACP1 P24666 3/20 0.46
APP P05067 1/20 0.45
ABL1 P00519 1/20 0.44
VNN1 O95497 2/20 0.43
USP2 O75604 1/20 0.42
ALDH1A1 P00352 1/20 0.42
LMNA P02545 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
TSHR P16473 1/20 0.42
MAPK1 P28482 1/20 0.42
CYP2C19 P33261 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30362451 0.83 CASR (0.46) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL19878225 0.83 CASR (0.46) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL30362764 0.82 CLK4 (0.44) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL19878451 0.82 CLK4 (0.44) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL5823848 0.79 APP (0.60) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL5494839 0.73 FGFR1 (0.52) CLK4ACP1ABL1USP2ALDH1A1
SCHEMBL29498169 0.72 RIPK2 (0.65) ABL1
SCHEMBL18571985 0.70 MEN1 (0.52) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL29911298 0.70 MEN1 (0.52) CLK4DYRK1ADYRK1BCLK1CLK2
SCHEMBL2805624 0.69 FGFR1 (0.44) CLK4DYRK1ADYRK1BCLK1CLK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109843858-A Certain chemical entities, composition and method 润新生物公司 2019-06-04 CN disclosed